Carbetocin Acetate
順序: Butyryl-Tyr(Me)-Ile-Gln-Asn-Cys-Pro-Leu-Gly-NH2 (Sulfide bond between Butyryl-4-yl and Cys)
CAS: 37025-55-1
外観: 白い粉
EINECS: 253-312-6
M.F.: C45H69N11O12S
M.W.: 988.17
Specific Optical Rotation D(c=1,1%HAc): -38.0~-42.0°
含水量(カール・フィッシャー): ≤5.0%
アセテート含有量(HPLCによる): ≤12.0%
アミノ酸組成: 理論値の±10%
純度 (HPLCによる): ≧98.0%
単一の不純物(HPLCによる): ≤1.0%
ペプチド含有量(by N%): 80%以上
アッセイ(無水による, 無酢酸 ): 97.0~103.0%
細菌エンドトキシン: ≤5EU/mg
使用法:An obstetric drug used to control postpartum hemorrhaging.
Carbetocin (宿, 禁止) (brand names Duratocin, Pabal, Lonactene, Depotocin, Comoton, Decomoton), or 1-butanoic acid-2-(O-methy-L-tyrosine)-1-carbaoxytocin, is an oxytocic used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section. It is an eight amino acid long analogue of oxytocin (a nonapeptide) そして, in accordance, has a similar action. Carbetocin primarily agonizes peripherally expressed oxytocin receptors.
Carbetocin is an oxytocic used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section. It is an eight amino acid long analogue of oxytocin (a nonapeptide) そして, in accordance, has a similar action. Carbetocin primarily agonizes peripherally expressed oxytocin receptors.