Produktnavn:Taltirelinacetat
Andre navn:PER-0910 Acetat;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (PER-0910 acetat) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| Molekylær formel: |
C17H31N7O9 |
| Molekylær vekt: |
477.46 |
| CAS-nr.: |
103300-74-9 |
| Utseende: |
hvitt pulver |
| Peptidinnhold(av %N): |
≥80 % |
| Acetatinnhold(ved HPLC): |
≤15% |
| Renhet(ved HPLC): |
0.98 |
| Enkel Urenhet(ved HPLC): |
≤1,0 % |
| Assay(Av vannfri, Eddiksyrefri): |
95.0~105,0 % |
| MS: |
Konsistent |
