productnaam:Taltireline-acetaat
Andere naam:PER-0910 Acetaat;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (PER-0910 acetaat) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| Moleculaire formule: |
C17H31N7O9 |
| Molecuulgewicht: |
477.46 |
| CAS-nr.: |
103300-74-9 |
| Uiterlijk: |
wit poeder |
| Peptide-inhoud(door %N): |
≥80% |
| Acetaat inhoud(door HPLC): |
≤15% |
| Zuiverheid(door HPLC): |
0.98 |
| Enkele onzuiverheid(door HPLC): |
≤1.0% |
| Assay(door watervrij, Azijnzuurvrij): |
95.0~105,0% |
| MEVROUW: |
Consequent |
