Produktname:Taltirelinacetat
Anderer Name:PRO-0910 Acetat;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (PRO-0910 Acetat) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| Molekularformel: |
C17H31N7Ö9 |
| Molekulargewicht: |
477.46 |
| CAS-Nr.: |
103300-74-9 |
| Aussehen: |
weißes Puder |
| Peptidgehalt(von %N): |
≥80% |
| Acetatgehalt(durch HPLC): |
≤15% |
| Reinheit(durch HPLC): |
0.98 |
| Einzelne Verunreinigung(durch HPLC): |
≤1,0 % |
| Probe(Von wasserfrei, Essigsäurefrei): |
95.0~105,0 % |
| FRAU: |
Konsistent |
