Product Name:Taltirelin Acetate
Other Name:TA-0910 Acetate;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
Molecular Formula: |
C17H31N7O9 |
Molecular Weight: |
477.46 |
CAS No.: |
103300-74-9 |
Appearance: |
White powder |
Peptide Content(by %N): |
≥80% |
Acetate Content(by HPLC): |
≤15% |
Purity(by HPLC): |
0.98 |
Single Impurity(by HPLC): |
≤1.0% |
Assay(By Anhydrous, Acetic Acid-free): |
95.0~105.0% |
MS: |
Consistent |