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Active Pharmaceuticals

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Product Name:Telapristone

Synonyma:Cdb 4124;proellex;telapristone (acetate);jvbgzfrptrksbb-mjbqoybxsa-n

CAS:198414-31-2 / 198414-30-1

MF:C31H39NO5

MW:505.64506

Telapristone (TABERNA), as telapristone acetate (proposed brand names Proellex, Progenta; former code name CDB-4124), Est synthetica, steroidal selective progesterone receptor modulator (SPRM) related to mifepristone which is under development by Repros Therapeutics for the treatment of breast cancer, endometriosis, and uterine fibroids.It was originally developed by the National Institutes of Health (NIH), et, as of 2017, is in phase II clinical trials for the aforementioned indications.In addition to its activity as an SPRM, the drug also has some antiglucocorticoid activity.

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