Mestanolone is the C-17 alpha alkylated version of DHT. This, of course, makes it orally bioavailable. It also adds some progestational activity to the molecule1. Methyl DHT cannot convert to estrogen, but it does bind strongly to SHBG which can displace estrogen into circulation possibly resulting in estrogenic side effects. As stated, DHT is deactivated in skeletal muscle by 3-alpha hydroxysteroid dehydrogenase as will Mestanolone.
Ermalone, a.k.a. methyldihydrotestosterone, mestanolone, and methyl-DHT is a modified version of dihydrotestosterone (DHT), an anabolic steroid that was designed to treat testosterone deficiency in males. Its c-17alpha alkylated modification allows it safe passage through the liver – the body’s primary filter for everything that’s orally ingested.
Since no further structural modification was added to protect the 3-ketone group, Ermalone is rapidly broken down within skeletal muscle tissue by the 3-alpha hydroxysteroid dehydrogenase enzyme. As a consequence, this oral androgen has an activity profile very similar to other non-aromatizing DHT-derived steroids like Winstrol and Oral Turinabol.
Mestanolone is perfect for reducing water weight gain, hardens muscles and leans out the muscle tissue throughout the body. It is the perfect toner and enhancer for any bodybuilder or serious weightlifter. It can be stacked with other products for the perfect cutting cycle pre-competition. It makes it that much easier to bulk up, maintain muscle mass and reduce unneeded weight. Mestanolone is used to:
- Increase testosterone benefit;
- Suppress estrogen effect;
- Lean muscle tissue;
- Increase strength;
- Improve drive and focus.